Iron-Catalyzed Synthesis of α-Dienyl Five- and Six-Membered N-Heterocycles
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چکیده
منابع مشابه
Intramolecular Pd(II)-catalyzed aerobic oxidative amination of alkenes: synthesis of six-membered N-heterocycles.
Use of a base-free Pd(DMSO)(2)(TFA)(2) catalyst system enables the synthesis of six-membered nitrogen heterocycles via a Wacker-type aerobic oxidative cyclization of alkenes bearing tethered sulfonamides. Various heterocycles, including morpholines, piperidines, piperazines, and piperazinones, are accessible by this method.
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ژورنال
عنوان ژورنال: European Journal of Organic Chemistry
سال: 2017
ISSN: 1434-193X
DOI: 10.1002/ejoc.201700977